SCHEMBL4714017

SCHEMBL4714017

CCc1c(N2CC[C@@H]([C@H](C)N)C2)c(F)cc2c(=O)n(N)c(=O)n(C3CC3)c12

nearest known ligand 0.79

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.53
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
CACNA1C Q13936 1/20 0.51
SCN5A Q14524 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4714018 1.00 KCNH2 (0.53) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4564657 1.00 KCNH2 (0.53) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1383199 0.89 KCNH2 (0.65) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1382157 0.89 KCNH2 (0.65) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1382153 0.89 KCNH2 (0.65) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4513751 0.89 KCNH2 (0.65) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4519616 0.89 KCNH2 (0.65) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4519620 0.89 KCNH2 (0.65) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4509668 0.88 KCNH2 (0.60) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4509664 0.88 KCNH2 (0.60) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255739-B1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER LAMBERT CO (US) 2008-06-11 EP claimed