SCHEMBL4714538

SCHEMBL4714538

O=C(Nc1ccc(F)cc1F)c1ccc(-c2cnc3ccc(-c4cn[nH]c4)cn23)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
ROCK2 O75116 4/20 0.41
ROCK1 Q13464 2/20 0.41
PIK3CA P42336 3/20 0.40
MTOR P42345 3/20 0.40
PIK3CD O00329 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
KIT P10721 1/20 0.39
FLT3 P36888 2/20 0.39
NRAS P01111 1/20 0.39
PTK6 Q13882 1/20 0.39
EPHB3 P54753 1/20 0.38
ERN1 O75460 1/20 0.38
MAPT P10636 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3848593 0.99 KDM4E (0.41) KDM4EHSD17B10RXFP1ROCK2ROCK1
SCHEMBL4712318 0.92 KDM4E (0.41) KDM4EHSD17B10RXFP1ROCK2ROCK1
Hydrochloric Acid SCHEMBL3849122 0.91 KDM4E (0.40) KDM4EHSD17B10RXFP1ROCK2ROCK1
Hydrochloric Acid SCHEMBL3846953 0.86 KIT (0.39) KDM4EROCK2ROCK1KITFLT3
Hydrochloric Acid SCHEMBL3850563 0.86 FLT3 (0.41) ROCK2ROCK1KITFLT3NRAS
SCHEMBL3848474 0.86 KDM4E (0.52) KDM4EHSD17B10RXFP1PIK3CAMTOR
Hydrochloric Acid SCHEMBL3852537 0.85 FLT3 (0.43) ROCK2ROCK1FLT3NRASPTK6
SCHEMBL3322932 0.85 KDM4E (0.46) KDM4EROCK2ROCK1KITFLT3
Hydrochloric Acid SCHEMBL3846069 0.84 KDM4E (0.46) KDM4EROCK2ROCK1KITFLT3
Hydrochloric Acid SCHEMBL3845647 0.81 LRRK2 (0.45) KDM4EROCK2ROCK1FLT3NRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP claimed