SCHEMBL4714740

SCHEMBL4714740

Nc1ccc2c(n1)NCCS2

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
RYR2 Q92736 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4714738 0.78 MEN1 (0.39) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL2800209 0.74 CCR1 (0.37) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL12692898 0.74 MEN1 (0.36) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL14610993 0.73 KDM4E (0.37) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL2051657 0.69 GAA (0.50) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL5760469 0.69 MEN1 (0.41) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL5298418 0.68 RYR2 (0.39) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL910393 0.67 MEN1 (0.39) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL15691803 0.66 UHRF1 (0.35) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL8168165 0.64 ITGAV (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216230-B1 FUSED CYCLOHEPTANE AND FUSED AZACYCLOHEPTANE COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR ANTAGONISTS AMGEN INC (US) 2008-04-23 EP disclosed