SCHEMBL4715033

SCHEMBL4715033

[CH2]Cc1ccc(C(=O)Nc2ccccc2N)cc1

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 18/20 0.70
HDAC2 Q92769 10/20 0.70
HDAC3 O15379 9/20 0.70
MAPK1 P28482 1/20 0.70
NCOR2 Q9Y618 3/20 0.68
PTGS1 P23219 1/20 0.63
HDAC4 P56524 3/20 0.63
HDAC7 Q8WUI4 3/20 0.63
HDAC10 Q969S8 3/20 0.63
HDAC11 Q96DB2 3/20 0.63
HDAC8 Q9BY41 3/20 0.63
HDAC6 Q9UBN7 3/20 0.63
HDAC9 Q9UKV0 3/20 0.63
HDAC5 Q9UQL6 3/20 0.63
NCOR1 O75376 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28155970 0.89 HDAC1 (0.64) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL8401704 0.88 HDAC1 (0.89) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL211677 0.87 HDAC1 (0.76) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL211107 0.87 HDAC1 (0.70) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL537019 0.87 HDAC1 (0.74) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL8470457 0.86 HDAC1 (0.68) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL2733350 0.86 HDAC1 (0.80) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL2732292 0.86 HDAC1 (0.70) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL4258366 0.83 HDAC1 (0.75) HDAC1HDAC2HDAC3MAPK1NCOR2
SCHEMBL8279067 0.83 HDAC1 (0.71) HDAC1HDAC2HDAC3MAPK1NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106966978-B Amide compound and preparation method and application thereof 北京化工大学 2020-06-26 CN disclosed
CN-106966978-A A kind of amides compound and its production and use 北京化工大学 2017-07-21 CN disclosed
EP-1904452-A2 HISTONE DEACETYLASE INHIBITORS Takeda San Diego, Inc. (US) 2008-04-02 EP disclosed
WO-2007011626-A2 HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2007-01-25 WO disclosed