SCHEMBL4716246

SCHEMBL4716246

CN1CCC(C(=O)Nc2cc(Oc3ccc(NC(=O)c4ccccc4N)c(Cl)c3)ccn2)CC1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRAF P15056 13/20 0.47
KDR P35968 15/20 0.47
MET P08581 3/20 0.47
KDM4E B2RXH2 1/20 0.46
NPC1 O15118 1/20 0.46
ALDH1A1 P00352 1/20 0.46
RAB9A P51151 1/20 0.46
RIPK1 Q13546 1/20 0.45
RIPK3 Q9Y572 1/20 0.45
AXL P30530 1/20 0.43
MERTK Q12866 1/20 0.43
FGFR1 P11362 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14540837 0.88 KDR (0.50) BRAFKDRMET
SCHEMBL14540841 0.85 BRAF (0.52) BRAFKDRMET
SCHEMBL1891544 0.83 KDR (0.58) BRAFKDR
SCHEMBL1891287 0.81 KDR (0.52) BRAFKDRRIPK3FGFR1
SCHEMBL4327777 0.80 BRAF (0.51) BRAFKDR
SCHEMBL1889996 0.79 KDR (0.61) BRAFKDR
SCHEMBL4335519 0.78 MEN1 (0.47) BRAFKDRMET
SCHEMBL4334102 0.77 KDR (0.51) BRAFKDRMETRIPK3
SCHEMBL4335858 0.76 KDR (0.58) BRAFKDR
SCHEMBL16037156 0.76 KDR (0.56) BRAFKDRMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506962-B1 Nitrogen-containing aromatic heterocycles EISAI R&D MAN CO LTD (JP) 2008-07-02 EP claimed