SCHEMBL471676

SCHEMBL471676

C=CO[C@H](C)[C@H]1[C@@H](/C=C/c2ccc(-c3cccc(F)c3)cn2)[C@@H]2CC[C@@H](NC(=O)OCC)C[C@H]2C[C@H]1C

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
F2R P25116 20/20 0.67
ABCB11 O95342 1/20 0.67
ADORA3 P0DMS8 1/20 0.67
CHRM1 P11229 1/20 0.67
SLC6A2 P23975 1/20 0.67
GPR183 P32249 1/20 0.67
OPRM1 P35372 1/20 0.67
KCNH2 Q12809 1/20 0.67
GPR35 Q9HC97 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14509113 0.82 F2R (0.80) F2RABCB11ADORA3CHRM1SLC6A2
SCHEMBL18597708 0.81 F2R (0.79) F2RABCB11ADORA3CHRM1SLC6A2
SCHEMBL1106148 0.81 F2R (0.76) F2RABCB11ADORA3CHRM1SLC6A2
SCHEMBL1106240 0.81 F2R (0.76) F2RABCB11ADORA3CHRM1SLC6A2
SCHEMBL16573430 0.81 F2R (0.70) F2RABCB11ADORA3CHRM1SLC6A2
SCHEMBL16901528 0.81 F2R (0.87) F2RABCB11ADORA3CHRM1SLC6A2
Vorapaxar SCHEMBL24988797 0.80 F2R (1.00) F2RABCB11ADORA3CHRM1SLC6A2
Vorapaxar SCHEMBL14203526 0.80 F2R (1.00) F2RABCB11ADORA3CHRM1SLC6A2
Vorapaxar SCHEMBL14203668 0.80 F2R (1.00) F2RABCB11ADORA3CHRM1SLC6A2
Vorapaxar SCHEMBL22122697 0.80 F2R (1.00) F2RABCB11ADORA3CHRM1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399912-A2 An exo-selective synthesis of himbacine analogs Schering Corporation (US) 2011-12-28 EP disclosed