SCHEMBL4717484

SCHEMBL4717484

Cc1cc(CC(NC(=O)ON2CCC(N3Cc4ccccc4NC3=O)CC2)C(=O)N2CCN(C3CCN(C)CC3)CC2)ccc1Br

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 18/20 0.56
CYP3A4 P08684 14/20 0.56
CALCA P06881 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719974 0.97 CALCRL (0.58) CALCRLCYP3A4CALCA
SCHEMBL4721310 0.94 CALCRL (0.52) CALCRLCYP3A4CALCA
SCHEMBL6226809 0.94 CALCRL (0.58) CALCRLCYP3A4
SCHEMBL4716556 0.93 CALCRL (0.64) CALCRLCYP3A4
SCHEMBL4717056 0.92 CALCRL (0.56) CALCRLCYP3A4
SCHEMBL4717363 0.91 CALCRL (0.56) CALCRLCYP3A4CALCA
SCHEMBL6223175 0.91 CALCRL (0.60) CALCRLCYP3A4
SCHEMBL3311366 0.90 CALCRL (0.68) CALCRLCYP3A4CALCA
SCHEMBL4718244 0.89 CALCRL (0.58) CALCRLCYP3A4
SCHEMBL6224283 0.89 CALCRL (0.57) CALCRLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558600-B1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2008-05-07 EP claimed
EP-1558600-B1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2008-05-07 EP disclosed