SCHEMBL4722763

SCHEMBL4722763

CS(=O)(=O)Nc1cc(Cl)c(-n2nc(-c3cc(Br)cc(-c4cnco4)c3)c3cccnc3c2=O)c(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 2/20 0.33
PFKFB3 Q16875 1/20 0.33
PFKFB4 Q16877 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
MET P08581 1/20 0.32
GLO1 Q04760 2/20 0.32
CKS1B P61024 1/20 0.32
SKP2 Q13309 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
BRD4 O60885 2/20 0.31
WDR5 P61964 1/20 0.31
JAK2 O60674 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720610 0.91 MEN1 (0.33) CCR9MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL4723380 0.88 BRAF (0.34) CCR9CKS1BSKP2MEN1KMT2A
SCHEMBL4723485 0.87 MEN1 (0.39) CYP2D6MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL4722898 0.86 MEN1 (0.35) MEN1KMT2AHPGDSMN1; SMN2NPSR1
SCHEMBL4723628 0.86 MEN1 (0.36) CCR9MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL4722814 0.84 MEN1 (0.36) CCR9CYP2D6MEN1KMT2AJAK2
SCHEMBL4719533 0.83 PDE4A (0.38) MEN1KMT2AHPGDSMN1; SMN2NPSR1
SCHEMBL4721827 0.80 PDE4A (0.35) CCR9PFKFB3PFKFB4MEN1KMT2A
SCHEMBL4723938 0.80 MEN1 (0.34) CCR9MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL4720482 0.80 MEN1 (0.34) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed