SCHEMBL4722917

SCHEMBL4722917

COc1cc(OC)cc(-c2nn(-c3cc(NCCCC(=O)N(C)C)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.33
MAPT P10636 3/20 0.33
TP53 P04637 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 2/20 0.33
CYP2C9 P11712 1/20 0.33
GRIA2 P42262 1/20 0.33
SCD O00767 1/20 0.33
TSHR P16473 2/20 0.33
NPY5R Q15761 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
SLC16A3 O15427 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721347 0.95 PDE4A (0.34) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4765721 0.92 PDE4A (0.36) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4719449 0.92 PDE4A (0.36) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4720140 0.92 PDE4A (0.37) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4723187 0.91 MAPT (0.34) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4722253 0.90 PDE4A (0.35) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4723364 0.90 PDE4A (0.35) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4721242 0.90 RAD52 (0.38) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4719833 0.90 PDE4A (0.35) SMN1; SMN2MAPTTP53PDE4APDE4B
SCHEMBL4718769 0.89 SCD (0.40) SMN1; SMN2MAPTTP53PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed