SCHEMBL4724734

SCHEMBL4724734

O=C(O)Cc1csc(-c2cc(Cl)ccc2OCc2ccccc2)n1

nearest known ligand 0.84

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 15/20 0.84
TBXA2R P21731 4/20 0.57
SHMT1 P34896 1/20 0.52
SHMT2 P34897 1/20 0.52
KMT2A Q03164 1/20 0.50
CYP2C9 P11712 1/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5129623 0.94 PTGER1 (0.75) PTGER1TBXA2RSHMT1SHMT2KDM4E
SCHEMBL4721023 0.90 PTGER1 (0.70) PTGER1TBXA2RSHMT1SHMT2CYP2C9
SCHEMBL14098698 0.89 PTGER1 (0.78) PTGER1TBXA2RSHMT1SHMT2KMT2A
SCHEMBL5121721 0.88 PTGER1 (0.67) PTGER1TBXA2RSHMT1SHMT2KDM4E
SCHEMBL4723494 0.87 PTGER1 (0.74) PTGER1TBXA2RKMT2ACYP2C9
SCHEMBL5125104 0.87 PTGER1 (0.66) PTGER1TBXA2RSHMT1SHMT2KDM4E
SCHEMBL5117064 0.87 PTGER1 (0.64) PTGER1CYP2C9KDM4EALDH1A1GAA
SCHEMBL5119199 0.86 PTGER1 (0.64) PTGER1SHMT1SHMT2CYP2C9KDM4E
SCHEMBL5115968 0.84 PTGER1 (0.61) PTGER1TBXA2RSHMT1SHMT2CYP2C9
SCHEMBL5129850 0.83 PTGER1 (0.60) PTGER1TBXA2RSHMT1SHMT2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080207708-A1 Oxazole and Thiazole Compounds and Their Use in the Treatment of Pge2 Mediated Disorders GLAXO GROUP LIMITED (GB) 2008-08-28 US disclosed
US-20080207708-A1 Oxazole and Thiazole Compounds and Their Use in the Treatment of Pge2 Mediated Disorders GLAXO GROUP LIMITED (GB) 2008-08-28 US disclosed
US-20080207708-A1 Oxazole and Thiazole Compounds and Their Use in the Treatment of Pge2 Mediated Disorders GLAXO GROUP LIMITED (GB) 2008-08-28 US disclosed
EP-1874776-A1 OXAZOLE AND THIAZOLE COMPOUNDS AND THEIR USE IN THE TREATMENT OF PGE2 MEDIATED DISORDERS GLAXO GROUP LIMITED (GB) 2008-01-09 EP disclosed
WO-2006114274-A1 OXAZOLE AND THIAZOLE COMPOUNDS AND THEIR USE IN THE TREATMENT OF PGE2 MEDIATED DISORDERS GLAXO GROUP LIMITED (GB) 2006-11-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080207708-A1 Oxazole and Thiazole Compounds and Their Use in the Treatment of Pge2 Mediated Disorders PTGER1, PTGER2, PTGER4 PTGER1 1/4885TBXA2R 10/4885SHMT1 2723/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.