SCHEMBL4725705

SCHEMBL4725705

NC(=O)CNCc1ccc2ccccc2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.51
HDAC2 Q92769 3/20 0.51
HDAC8 Q9BY41 3/20 0.51
HDAC6 Q9UBN7 1/20 0.51
CYP1A2 P05177 1/20 0.48
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
ADORA2A P29274 2/20 0.44
ADORA1 P30542 1/20 0.44
KDM4C Q9H3R0 1/20 0.43
GPBAR1 Q8TDU6 2/20 0.43
KDM1A O60341 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
FAAH O00519 1/20 0.41
MGAM O43451 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8843274 0.86 KDM4C (0.55) HDAC1HDAC2HDAC8HDAC6CYP1A2
Hydrochloric Acid SCHEMBL8843524 0.84 KDM4C (0.54) HDAC1HDAC2HDAC8HDAC6CYP1A2
SCHEMBL24943587 0.81 HDAC1 (0.55) HDAC1HDAC2HDAC8HDAC6CYP1A2
SCHEMBL12749489 0.79 CYSLTR2 (0.54) HDAC1HDAC2HDAC8HDAC6CYP1A2
SCHEMBL5503169 0.78 CYP1A2 (0.63) HDAC1HDAC2CYP1A2ALDH1A1GAA
SCHEMBL29877127 0.78 CYP1A2 (0.63) HDAC1HDAC2CYP1A2ALDH1A1GAA
SCHEMBL30388584 0.78 KDM1A (0.50) HDAC1HDAC2HDAC8HDAC6CYP1A2
SCHEMBL10616742 0.76 KDM1A (0.49) HDAC1HDAC2HDAC8HDAC6CYP1A2
SCHEMBL15578063 0.76 HDAC1 (0.61) HDAC1HDAC2HDAC8HDAC6CYP1A2
SCHEMBL1037883 0.76 HDAC1 (0.48) HDAC1HDAC2HDAC8HDAC6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021745-A2 HEPATITIS C VIRUS ENTRY INHIBITORS ITHERX PHARMACEUTICALS, INC. (US) 2008-02-21 WO disclosed
US-6399631-B1 3-AMIDO OR 3-SULFONAMIDO; EATING DISORDERS IN HUMANS, DOGS AND CATS PFIZER INC. 2002-06-04 US disclosed
US-5672615-A MATRIX-DEGRADING METALLOPROTEINASE INHIBITORS NOVARTIS CORPORATION (US) 1997-09-30 US disclosed