SCHEMBL4726802

SCHEMBL4726802

S=C(Nc1cccc(Cl)c1)NC1CCN(c2ncnc3cc(Cl)ccc23)CC1.S=C(Nc1ccccc1)NC1CCN(c2ncnc3cc(Cl)ccc23)CC1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 1/20 0.54
CYP1A2 P05177 2/20 0.53
CYP2D6 P10635 2/20 0.53
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C19 P33261 1/20 0.52
PDGFRB P09619 3/20 0.52
LMNA P02545 2/20 0.47
ALDH1A1 P00352 2/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4582925 0.97 PAK1 (0.57) PAK1CYP1A2CYP2D6KMT2AMEN1
SCHEMBL4584207 0.96 CYP1A2 (0.56) PAK1CYP1A2CYP2D6KMT2AMEN1
SCHEMBL4582847 0.90 CYP1A2 (0.52) PAK1CYP1A2CYP2D6KMT2AMEN1
SCHEMBL4583131 0.88 PDGFRB (0.53) PAK1CYP1A2CYP2D6PDGFRBALDH1A1
SCHEMBL4582263 0.88 CYP1A2 (0.49) PAK1CYP1A2CYP2D6KMT2AMEN1
SCHEMBL4583185 0.88 CYP1A2 (0.49) PAK1CYP1A2CYP2D6KMT2AMEN1
SCHEMBL4584940 0.87 CYP1A2 (0.54) PAK1CYP1A2CYP2D6CYP3A4CYP2C19
SCHEMBL4726373 0.86 CYP1A2 (0.46) PAK1CYP1A2CYP2D6KMT2AMEN1
SCHEMBL4728704 0.86 EGFR (0.46) PAK1CYP1A2CYP2D6KMT2AMEN1
SCHEMBL4583789 0.85 PAK1 (0.49) PAK1CYP1A2CYP2D6KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008028690-A1 1-(HET)ARYL-3-[HETARYL-PIPERIDIN-4-YL]-THIOUREAS AS MODULATORS OF THE EP2 RECEPTOR BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-03-13 WO disclosed