SCHEMBL4728279

SCHEMBL4728279

NNC(=O)c1ccc2cncc(Br)c2n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.47
P2RX7 Q99572 4/20 0.45
KDM4E B2RXH2 3/20 0.41
CCNC P24863 5/20 0.40
CDK8 P49336 5/20 0.40
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
OGG1 O15527 1/20 0.36
MPO P05164 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2C19 P33261 1/20 0.36
HDAC8 Q9BY41 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4579695 0.84 CCNC (0.52) CCNCCDK8HDAC8NPC1
SCHEMBL15742867 0.84 CNR1 (0.39) ALDH1A1MAPTKDM4ECCNCCDK8
SCHEMBL1319809 0.82 CCNC (0.49) CCNCCDK8ADORA3
SCHEMBL15741600 0.80 CCNC (0.38) ALDH1A1CCNCCDK8
SCHEMBL15742716 0.80 SCN9A (0.43) CCNCCDK8
SCHEMBL29850571 0.80 CCNC (0.47) ALDH1A1MAPTKDM4ECCNCCDK8
SCHEMBL578828 0.80 CCNC (0.47) ALDH1A1MAPTKDM4ECCNCCDK8
SCHEMBL4580627 0.80 SMYD3 (0.42) CCNCCDK8
SCHEMBL15742739 0.79 HPGD (0.55) ALDH1A1MAPTKDM4ECYP1A2NPC1
SCHEMBL15742746 0.79 SMN1; SMN2 (0.52) ALDH1A1GAAHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith D SIDOCKY NEIL R 2008-10-02 US disclosed
WO-2008036308-A2 AMINO-SUBSTITUTED HETEROCYCLES, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2008-03-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith JAK2, CHEK2, MTOR ALDH1A1 1752/4885MAPT 4243/4885GAA 2251/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.