SCHEMBL473000

SCHEMBL473000

CCC(C(=O)O)n1nnc(-c2coc(N3CCC(Oc4cc(F)ccc4Br)CC3)n2)n1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCD O00767 17/20 0.49
SCD5 Q86SK9 1/20 0.45
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473021 0.87 SCD (0.46) SCDSCD5
SCHEMBL473023 0.87 SCD (0.54) SCDSCD5KDM4EALDH1A1HPGD
SCHEMBL472987 0.85 SCD (0.68) SCDSCD5
SCHEMBL27889871 0.83 SCD (0.48) SCDSCD5
SCHEMBL27765338 0.83 SCD (0.47) SCDSCD5
SCHEMBL473052 0.82 SCD (0.73) SCDSCD5
SCHEMBL473059 0.81 SCD (0.73) SCDSCD5KDM4EALDH1A1HPGD
SCHEMBL3020613 0.77 SCD (0.62) SCDSCD5
SCHEMBL473054 0.77 SCD (0.51) SCDSCD5ALDH1A1HPGD
SCHEMBL12130242 0.77 SCD (0.55) SCDSCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099793-B1 AZACYCLOALKANE DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK CANADA INC (CA) 2012-02-01 EP disclosed
US-8063224-B2 [5-(5-{4-[2-(Trifluoromethyl)phenoxy]piperidin-1-yl}-1,3,4-thiadiazol-2-yl)-2H-tetrazol-2-yl]acetic acid; metabolic disorders,antidiabetic, hypoglycemic agent; obesity, insulin resistance, liver steatosis, atherosclerosis, neurological disease, dyslipidemia, hyperlipidemia, low HDL, and high LDL MERCK CANADA INC. (CA) 2011-11-22 US disclosed