SCHEMBL4733802

SCHEMBL4733802

CCOc1cnc(NC(=O)C2(CC)CCCC2)cc1CN1CCOCC1

nearest known ligand 0.76

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 11/20 0.76
CNR1 P21554 5/20 0.76
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
SAE1 Q9UBE0 1/20 0.40
UBA2 Q9UBT2 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TSHR P16473 1/20 0.39
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
CHEK1 O14757 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4733039 0.99 CNR2 (0.77) CNR2CNR1LMNAMAPTCACNA1B
SCHEMBL4732125 0.98 CNR2 (0.76) CNR2CNR1LMNAMAPTCACNA1B
SCHEMBL4734621 0.92 CNR2 (0.76) CNR2CNR1KDM4EALDH1A1PDCD1
SCHEMBL4732582 0.91 CNR2 (0.77) CNR2CNR1KDM4EALDH1A1PDCD1
SCHEMBL4732648 0.90 CNR2 (0.76) CNR2CNR1LMNAMAPTKDM4E
SCHEMBL4729957 0.88 CNR2 (0.60) CNR2CNR1LMNAMAPTCACNA1B
SCHEMBL4732972 0.88 CNR2 (0.82) CNR2CNR1TSHRPDCD1CD274
SCHEMBL4732987 0.87 CNR2 (1.00) CNR2CNR1PDCD1CD274
SCHEMBL4732822 0.87 CNR2 (0.83) CNR2CNR1PDCD1CD274
SCHEMBL4732451 0.86 CNR2 (1.00) CNR2CNR1PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO claimed
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed