SCHEMBL4735167

SCHEMBL4735167

Cc1ccc(-c2c(N(C)C(=O)O)c(CC3CC3)nc3ccc(O)cc23)cc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 11/20 0.38
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
ESRRB O95718 1/20 0.36
ESRRA P11474 1/20 0.36
MELK Q14680 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3901983 0.84 DPP4 (0.41) DPP4ESR1ESR2ESRRBESRRA
SCHEMBL3892488 0.84 DPP4 (0.52) DPP4
SCHEMBL3903159 0.80 DPP4 (0.41) DPP4
SCHEMBL3893787 0.79 ESRRB (0.41) DPP4GRIN1GRIN2BESR1ESR2
SCHEMBL4708341 0.78 DPP4 (0.38) DPP4GRIN1GRIN2B
SCHEMBL4708340 0.77 GRIN1 (0.36) DPP4GRIN1GRIN2BESR1ESR2
SCHEMBL3902200 0.75 DPP4 (0.50) DPP4ESR1ESR2
SCHEMBL3895506 0.73 DPP4 (0.55) DPP4
SCHEMBL3907628 0.72 DPP4 (0.54) DPP4
SCHEMBL3897641 0.72 DPP4 (0.57) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1527049-B1 FUSED HETEROCYCLIC COMPOUNDS AS PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2008-07-16 EP disclosed