SCHEMBL4736846

SCHEMBL4736846

COc1cccc(Oc2nc(N)nc3c2-c2cc(S(=O)(=O)N4CCOCC4)c(Cl)cc2CC3)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CASP1 P29466 1/20 0.39
LMNA P02545 3/20 0.38
KMT2A Q03164 2/20 0.37
MAPT P10636 2/20 0.36
TYMS P04818 1/20 0.36
THRB P10828 1/20 0.36
POLB P06746 1/20 0.36
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739051 0.78 ADORA2A (0.48) KDM4ELMNAKMT2AMAPTPOLB
SCHEMBL4738561 0.78 TSHR (0.48) TSHRHSD17B10LMNAKMT2AMAPT
SCHEMBL14147957 0.77 ADORA2A (0.42) TSHRKDM4ELMNAKMT2AMAPT
SCHEMBL14147958 0.76 SMN1; SMN2 (0.42) TSHRKDM4EHSD17B10KMT2ATP53
SCHEMBL14147951 0.76 ALOX5AP (0.44) TSHRKDM4ELMNAMAPT
SCHEMBL14147954 0.75 ADORA2A (0.39) TSHRKDM4EHSD17B10KMT2AMAPT
SCHEMBL14147955 0.75 ADORA2A (0.46) KDM4EKMT2AMAPTTDP1
SCHEMBL14147950 0.74 MEN1 (0.40) KDM4ELMNAKMT2AMAPTMTOR
SCHEMBL14147952 0.73 BRAF (0.45) KDM4ELMNAKMT2AMAPTPOLB
SCHEMBL14147959 0.73 MAPT (0.43) TSHRKDM4EHSD17B10LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed