SCHEMBL4737873

SCHEMBL4737873

O=C(O)c1cc(F)c(N2CCC(C(=O)NS(=O)(=O)Cc3ccccc3)CC2)nc1CN1CCCC1=O

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 16/20 0.50
CYP3A4 P08684 5/20 0.48
CYP2C9 P11712 6/20 0.47
CHRM2 P08172 1/20 0.47
DRD3 P35462 1/20 0.47
STS P08842 1/20 0.42
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4172600 0.91 P2RY12 (0.63) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4737184 0.91 P2RY12 (0.49) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4737254 0.91 P2RY12 (0.58) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4852691 0.89 P2RY12 (0.52) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4740631 0.89 P2RY12 (0.64) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4737929 0.86 P2RY12 (0.63) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4175823 0.83 P2RY12 (0.63) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4171008 0.83 P2RY12 (0.64) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4170985 0.82 P2RY12 (0.61) P2RY12CYP3A4CYP2C9CHRM2DRD3
SCHEMBL4737218 0.82 P2RY12 (0.58) P2RY12CYP3A4CYP2C9CHRM2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008085119-A1 NEW PYRIDINE ANALOGUES VIII 518 ASTRAZENECA AB (SE) 2008-07-17 WO disclosed