SCHEMBL4740253

SCHEMBL4740253

COc1cc2ncnc(NCCc3ccc(Cl)cc3)c2cc1OCCCCCCC(=O)NO

nearest known ligand 0.84

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.84
HDAC3 O15379 16/20 0.75
HDAC4 P56524 16/20 0.75
HDAC1 Q13547 16/20 0.75
HDAC7 Q8WUI4 16/20 0.75
HDAC2 Q92769 16/20 0.75
HDAC10 Q969S8 16/20 0.75
HDAC11 Q96DB2 16/20 0.75
HDAC8 Q9BY41 16/20 0.75
HDAC6 Q9UBN7 16/20 0.75
HDAC9 Q9UKV0 16/20 0.75
HDAC5 Q9UQL6 16/20 0.75
KDR P35968 12/20 0.75
ERBB2 P04626 5/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739400 0.92 EGFR (0.85) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL13058955 0.91 HDAC3 (0.84) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL3643141 0.91 EGFR (0.72) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL4740648 0.91 EGFR (1.00) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL4737117 0.91 EGFR (1.00) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL641614 0.84 ERBB2 (1.00) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL3649149 0.83 EGFR (0.73) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL13059538 0.83 HDAC3 (0.85) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL27926496 0.83 EGFR (0.72) EGFRHDAC3HDAC4HDAC1HDAC7
SCHEMBL3649079 0.83 EGFR (0.85) EGFRHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033747-A9 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS CURIS INC (MA) 2008-07-24 WO disclosed