SCHEMBL4742763

SCHEMBL4742763

CCCC(C)(CC(=O)O)CC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.48
CHRM1 P11229 1/20 0.48
TBXA2R P21731 1/20 0.48
ADRA1A P35348 1/20 0.48
FFAR1 O14842 1/20 0.46
CPT2 P23786 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
CYP2C19 P33261 2/20 0.46
HIF1A Q16665 2/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
LMNA P02545 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KDM4E B2RXH2 1/20 0.41
FFAR3 O14843 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HSPD1 P10809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5540263 0.95 HMGCR (0.48) HMGCRCHRM1TBXA2RADRA1AFFAR1
SCHEMBL11922837 0.90 HMGCR (0.44) HMGCRCHRM1TBXA2RADRA1AFFAR1
SCHEMBL15237487 0.86 TDP1 (0.45) HMGCRCHRM1TBXA2RADRA1AFFAR1
SCHEMBL31021331 0.85 TDP1 (0.48) HMGCRCHRM1TBXA2RADRA1AFFAR1
SCHEMBL2349178 0.80 TDP1 (0.48) HMGCRCHRM1TBXA2RADRA1AFFAR1
SCHEMBL544642 0.80 HMGCR (0.61) HMGCRCHRM1TBXA2RADRA1AFFAR1
SCHEMBL974936 0.79 FFAR1 (0.65) HMGCRCHRM1TBXA2RADRA1AFFAR1
SCHEMBL10776763 0.78 TDP1 (0.52) FFAR1CPT2TDP1TSHRHSD17B10
SCHEMBL18850502 0.78 FFAR1 (0.47) HMGCRCHRM1TBXA2RADRA1AFFAR1
SCHEMBL1419066 0.78 HMGCR (0.52) HMGCRCHRM1TBXA2RADRA1AFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008099019-A1 6-HYDROXY-DIBENZODIAZEPINONES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed
WO-2008099019-A1 6-HYDROXY-DIBENZODIAZEPINONES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed