SCHEMBL4743428

SCHEMBL4743428

CCOC(=O)c1cnc2cc(C(Cl)(Cl)Cl)ccc2c1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
PDE5A O76074 2/20 0.49
PDE6D O43924 1/20 0.49
PDE6A P16499 1/20 0.49
PDE6G P18545 1/20 0.49
PDE6B P35913 1/20 0.49
PDE6C P51160 1/20 0.49
PDE6H Q13956 1/20 0.49
THRB P10828 2/20 0.48
MAPT P10636 6/20 0.48
GAA P10253 4/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPK10 P53779 1/20 0.47
MAPK1 P28482 2/20 0.45
CA2 P00918 1/20 0.43
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL263314 0.90 KMT2A (0.53) KMT2AMEN1PDE5APDE6DPDE6A
SCHEMBL429137 0.89 PDE5A (0.60) KMT2AMEN1PDE5APDE6DPDE6A
SCHEMBL12426321 0.85 KMT2A (0.57) KMT2AMEN1THRBMAPTGAA
SCHEMBL1178069 0.85 KMT2A (0.58) KMT2AMEN1THRBMAPTGAA
SCHEMBL4428236 0.84 PDE5A (0.56) KMT2AMEN1PDE5APDE6DPDE6A
SCHEMBL2723785 0.82 GAA (0.57) KMT2AMEN1THRBMAPTGAA
SCHEMBL621104 0.82 KMT2A (0.55) KMT2AMEN1PDE5APDE6DPDE6A
SCHEMBL1467397 0.81 KMT2A (0.54) KMT2AMEN1THRBMAPTGAA
SCHEMBL18987698 0.81 TP53 (0.54) KMT2AMEN1PDE5APDE6DPDE6A
SCHEMBL1285507 0.81 MAPT (0.51) KMT2AMEN1PDE5AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed