SCHEMBL4744236

SCHEMBL4744236

O=C(NCc1ccnc2ccccc12)c1cnc2cc(C(F)(F)F)c(Cl)cc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
HPGDS O60760 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
KDR P35968 2/20 0.41
TP53 P04637 1/20 0.41
DDR1 Q08345 1/20 0.41
EPHX2 P34913 3/20 0.40
TACR1 P25103 1/20 0.40
PPARD Q03181 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
PSMD14 O00487 1/20 0.39
STAMBP O95630 1/20 0.39
KLKB1 P03952 1/20 0.39
MAP4K1 Q92918 1/20 0.39
CNR2 P34972 1/20 0.39
DGAT2 Q96PD7 1/20 0.39
FLT1 P17948 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739588 0.89 ADORA2A (0.48) ADORA2AADORA1HPGDSKDREPHX2
SCHEMBL14148289 0.84 TRPV1 (0.49) SMN1; SMN2TP53PSMD14STAMBPDGAT2
SCHEMBL4787180 0.76 FLT1 (0.48) ADORA2AADORA1SMN1; SMN2KDRTP53
SCHEMBL14147888 0.74 TRPV1 (0.49) SMN1; SMN2PSMD14STAMBPDGAT2
SCHEMBL1644237 0.71 EGLN1 (0.46) PSMD14
SCHEMBL269559 0.69 SMN1; SMN2 (0.49) ADORA2AADORA1SMN1; SMN2KDREPHX2
SCHEMBL263858 0.69 SMN1; SMN2 (0.43) ADORA2AADORA1SMN1; SMN2KDRDDR1
SCHEMBL14147908 0.68 SCN9A (0.52) ADORA2AADORA1KDRFLT1
SCHEMBL264360 0.68 SMN1; SMN2 (0.48) ADORA2AADORA1HPGDSSMN1; SMN2KDR
SCHEMBL14147719 0.67 TRPV1 (0.49) ADORA2AHPGDSTP53PPARDPSMD14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008090434-A1 SUBSTITUTED N-BICYCLICALKYL BICYCLIC CARBOXYAMIDE COMPOUNDS PFIZER JAPAN INC. (JP) 2008-07-31 WO claimed
WO-2008090434-A1 SUBSTITUTED N-BICYCLICALKYL BICYCLIC CARBOXYAMIDE COMPOUNDS PFIZER JAPAN INC. (JP) 2008-07-31 WO disclosed