SCHEMBL4744978

SCHEMBL4744978

CC(C)NC(=O)CN1CCN(CCCCOc2ccc3c(-c4ccc(Cl)cc4)coc3c2)CC1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.54
PDK1 Q15118 1/20 0.47
PDK2 Q15119 1/20 0.47
BCHE P06276 2/20 0.46
ACHE P22303 2/20 0.46
AVPR1B P47901 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742617 0.99 HRH3 (0.53) HRH3PDK1PDK2BCHEACHE
SCHEMBL4745561 0.99 HRH3 (0.53) HRH3PDK1PDK2BCHEACHE
SCHEMBL4745673 0.97 HRH3 (0.51) HRH3PDK1PDK2AVPR1B
SCHEMBL4745559 0.95 HRH3 (0.54) HRH3PDK1PDK2AVPR1B
SCHEMBL4746425 0.92 HRH3 (0.63) HRH3PDK1PDK2BCHEACHE
SCHEMBL4788438 0.91 HRH3 (0.49) HRH3PDK1PDK2BCHEACHE
SCHEMBL4746415 0.91 AVPR1B (0.53) HRH3PDK1PDK2AVPR1B
SCHEMBL4746404 0.91 HRH3 (0.50) HRH3PDK1PDK2BCHEACHE
SCHEMBL4742548 0.91 HRH3 (0.53) HRH3PDK1PDK2BCHEACHE
SCHEMBL4746377 0.91 HRH3 (0.53) HRH3BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107321-A1 HETEROCYCLIC COMPOUNDS USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO claimed
WO-2008107321-A1 HETEROCYCLIC COMPOUNDS USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed