SCHEMBL4745252

SCHEMBL4745252

CC(N)C(N)Cc1cc(F)cc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.40
DPP4 P27487 1/20 0.38
TRPA1 O75762 1/20 0.34
NR3C1 P04150 1/20 0.33
PGR P06401 1/20 0.33
NR3C2 P08235 1/20 0.33
CYP2D6 P10635 1/20 0.33
EPHX1 P07099 1/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 1/20 0.32
SMYD3 Q9H7B4 1/20 0.31
TAAR1 Q96RJ0 2/20 0.31
MAOA P21397 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17407620 0.87 DPP4 (0.52) IDO1DPP4TRPA1NR3C1PGR
SCHEMBL14478271 0.82 SLC6A2 (0.48) HTR2AHTR2CHTR2BTAAR1MAOA
SCHEMBL14478296 0.82 SLC6A2 (0.48) HTR2AHTR2CHTR2BTAAR1MAOA
SCHEMBL17413330 0.82 SLC6A2 (0.48) HTR2AHTR2CHTR2BTAAR1MAOA
SCHEMBL2623872 0.77 IDO1 (0.41) IDO1TRPA1NR3C1PGRNR3C2
SCHEMBL19737292 0.74 IDO1 (0.40) IDO1DPP4TRPA1NR3C1PGR
SCHEMBL13814727 0.74 IDO1 (0.36) IDO1DPP4EPHX1SLC6A2SLC6A4
SCHEMBL4823652 0.74 IDO1 (0.36) IDO1DPP4TRPA1EPHX1
SCHEMBL4413267 0.73 IDO1 (0.38) IDO1TRPA1NR3C1PGRNR3C2
SCHEMBL9071082 0.73 IDO1 (0.38) IDO1TRPA1NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008109613-A1 BENZO[C][2,7]NAPHTHYRIDINE DERIVATIVES, AND THEIR USE AS KINASE INHIBITORS WYETH (US) 2008-09-12 WO disclosed