SCHEMBL4746288

SCHEMBL4746288

Clc1ccc(CN(C2CCCC2)C2CCNC2)c(Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 18/20 0.64
SLC6A2 P23975 16/20 0.64
NOS2 P35228 2/20 0.60
CYP2D6 P10635 5/20 0.59
KCNH2 Q12809 2/20 0.59
SLC6A3 Q01959 7/20 0.57
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
NOS3 P29474 1/20 0.47
NOS1 P29475 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4486154 1.00 SLC6A4 (0.64) SLC6A4SLC6A2NOS2CYP2D6KCNH2
SCHEMBL4485355 0.99 SLC6A4 (0.63) SLC6A4SLC6A2NOS2CYP2D6KCNH2
SCHEMBL4476276 0.89 SLC6A4 (0.67) SLC6A4SLC6A2CYP2D6KCNH2SLC6A3
SCHEMBL4483224 0.89 SLC6A4 (0.57) SLC6A4SLC6A2NOS2CYP2D6KCNH2
SCHEMBL4489382 0.87 SLC6A4 (0.57) SLC6A4SLC6A2NOS2CYP2D6KCNH2
SCHEMBL4489380 0.87 SLC6A4 (0.57) SLC6A4SLC6A2NOS2CYP2D6KCNH2
SCHEMBL4479763 0.84 SLC6A4 (0.64) SLC6A4SLC6A2NOS2CYP2D6KCNH2
SCHEMBL4499777 0.83 SLC6A2 (0.66) SLC6A4SLC6A2NOS2CYP2D6KCNH2
Cadaverine Tartrate SCHEMBL4477362 0.80 SLC6A4 (0.58) SLC6A4SLC6A2CYP2D6KCNH2SLC6A3
Cadaverine Tartrate SCHEMBL4486665 0.80 SLC6A2 (0.58) SLC6A4SLC6A2CYP2D6KCNH2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638934-B1 3-AMINOPYRROLIDINES AS INHIBITORS OF MONOAMINE UPTAKE LILLY CO ELI (US) 2008-01-09 EP disclosed
EP-1638934-A1 3-AMINOPYRROLIDINES AS INHIBITORS OF MONOAMINE UPTAKE ELI LILLY AND COMPANY (US) 2006-03-29 EP disclosed
WO-2005000811-A1 3-AMINOPYRROLIDINES AS INHIBITORS OF MONOAMINE UPTAKE ELI LILLY AND COMPANY (US) 2005-01-06 WO disclosed