SCHEMBL4746934

SCHEMBL4746934

O=C(O)N[C@@H]1COc2cccc(-c3ccncc3)c2C1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 19/20 0.66
KCNH2 Q12809 12/20 0.66
SCN5A Q14524 13/20 0.64
SLC6A3 Q01959 1/20 0.44
GHSR Q92847 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL840782 0.81 SCN9A (1.00) SCN9AKCNH2SCN5ASLC6A3GHSR
SCHEMBL841447 0.80 SCN9A (0.70) SCN9AKCNH2SCN5ASLC6A3GHSR
SCHEMBL841280 0.79 SCN9A (0.57) SCN9AKCNH2SCN5ASLC6A3GHSR
SCHEMBL839807 0.79 SCN9A (1.00) SCN9AKCNH2SCN5ASLC6A3GHSR
SCHEMBL841680 0.78 SCN9A (0.62) SCN9AKCNH2SCN5ASLC6A3GHSR
SCHEMBL20873473 0.78 SCN9A (0.42) SCN9AKCNH2SCN5A
SCHEMBL4747000 0.78 SCN9A (0.42) SCN9AKCNH2SCN5A
SCHEMBL840991 0.77 SCN9A (0.63) SCN9AKCNH2SCN5ASLC6A3GHSR
SCHEMBL840760 0.77 SCN9A (0.72) SCN9AKCNH2SCN5ASLC6A3GHSR
SCHEMBL839786 0.77 SCN9A (0.62) SCN9AKCNH2SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO claimed
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed