SCHEMBL474750

SCHEMBL474750

CC(C)CC(=O)N[C@H](C(=O)N1CCCC1C(=O)Nc1ccc2[nH]c(-c3ccc(NC(=O)[C@@H]4CCCN4C(=O)[C@H](NC(=O)CC(C)C)c4ccccc4)cc3)cc2c1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.57
CYP2C9 P11712 6/20 0.52
CYP2C19 P33261 6/20 0.52
CYP3A4 P08684 5/20 0.52
CYP2D6 P10635 2/20 0.52
CYP1A2 P05177 2/20 0.52
HCRTR1 O43613 3/20 0.43
HCRTR2 O43614 3/20 0.43
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
ALDH1A1 P00352 3/20 0.40
SLC2A1 P11166 1/20 0.40
MAPT P10636 1/20 0.39
GAA P10253 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
PABPC1 P11940 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22344978 1.00 KCNH2 (0.57) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL474751 1.00 KCNH2 (0.57) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL18379459 0.94 KCNH2 (0.52) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL895306 0.90 KCNH2 (0.56) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL10223645 0.88 KCNH2 (0.75) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL20952453 0.88 KCNH2 (0.60) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL16188351 0.88 KCNH2 (0.60) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL16188303 0.88 KCNH2 (0.60) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL20966484 0.88 KCNH2 (0.46) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL22344943 0.88 KCNH2 (0.59) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410844-A1 INHIBITORS OF HEPATITIS C VIRUS REPLICATION Merck Sharp & Dohme Corp. (US) 2012-02-01 EP claimed