SCHEMBL4748128

SCHEMBL4748128

CN1CCN(c2cccc3c2C[C@H](NC(=O)c2ccc(C(C)(C)C)cc2)CO3)CC1

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 9/20 0.75
KCNH2 Q12809 7/20 0.75
SCN5A Q14524 7/20 0.75
HTR2A P28223 7/20 0.47
DRD3 P35462 7/20 0.47
DRD2 P14416 6/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4841770 0.91 SCN9A (0.80) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL4830458 0.91 SCN9A (0.80) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL4830465 0.91 SCN9A (0.80) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL4830436 0.87 SCN9A (0.71) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL8075533 0.87 SCN9A (0.71) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL4836383 0.87 SCN9A (0.71) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL4838340 0.86 KCNH2 (0.70) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL4838380 0.86 KCNH2 (0.70) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL4838400 0.86 KCNH2 (0.70) SCN9AKCNH2SCN5AHTR2ADRD3
SCHEMBL4842018 0.86 KCNH2 (0.70) SCN9AKCNH2SCN5AHTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130322-A1 NOVEL 5-HETEROCYCLYL-CHROMANE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO claimed
WO-2008130322-A1 NOVEL 5-HETEROCYCLYL-CHROMANE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed