SCHEMBL4751745

SCHEMBL4751745

CC(=O)c1ccccc1Nc1ccnc2cc(Cl)ccc12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.62
ALDH1A1 P00352 3/20 0.62
CYP3A4 P08684 2/20 0.62
MAPK1 P28482 2/20 0.62
HSD17B10 Q99714 2/20 0.62
CYP2D6 P10635 2/20 0.62
HPGD P15428 2/20 0.62
KDM4E B2RXH2 2/20 0.62
MLNR O43193 1/20 0.62
ABCB11 O95342 1/20 0.62
CHRM2 P08172 1/20 0.62
ADORA3 P0DMS8 1/20 0.62
CHRM1 P11229 1/20 0.62
GABRA1 P14867 1/20 0.62
TBXA2R P21731 1/20 0.62
PTGS1 P23219 1/20 0.62
SLC6A2 P23975 1/20 0.62
PDE4A P27815 1/20 0.62
ADORA2A P29274 1/20 0.62
ADRA1A P35348 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL598101 0.89 CYP1A2 (0.65) CYP1A2ALDH1A1CYP3A4MAPK1HSD17B10
SCHEMBL10951691 0.88 CYP1A2 (0.64) CYP1A2ALDH1A1CYP3A4MAPK1HSD17B10
SCHEMBL10951705 0.88 CYP1A2 (0.64) CYP1A2ALDH1A1CYP3A4MAPK1HSD17B10
SCHEMBL10951695 0.86 CYP1A2 (0.61) CYP1A2ALDH1A1CYP3A4MAPK1HSD17B10
SCHEMBL21346898 0.85 CYP1A2 (0.63) CYP1A2ALDH1A1CYP3A4MAPK1HSD17B10
SCHEMBL21346880 0.84 DNMT1 (0.56) ADRA1AKMT2AMEN1
SCHEMBL21346888 0.84 KDM4E (0.73) CYP1A2ALDH1A1CYP3A4MAPK1HSD17B10
SCHEMBL11525169 0.81 CYP3A4 (0.69) CYP1A2ALDH1A1CYP3A4MAPK1HSD17B10
SCHEMBL21346896 0.81 KMT2A (0.60) CYP1A2ALDH1A1CYP3A4MAPK1HSD17B10
SCHEMBL21121619 0.80 POLB (0.67) CYP1A2ALDH1A1HPGDKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135886-A2 QUINOLINE DERIVATIVES FOR USE IN THE INHIBITION OF THE GROWTH OF TUMOUR CELLS UNIVERSITY OF PRETORIA (ZA) 2008-11-13 WO disclosed