SCHEMBL4752569

SCHEMBL4752569

CN1CCN(c2cc(NCCC3CC3)ncn2)CC1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 14/20 0.70
HRH3 Q9Y5N1 3/20 0.70
HRH2 P25021 1/20 0.70
KDR P35968 1/20 0.46
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
PIK3CB P42338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1775555 0.86 HRH4 (0.65) HRH4HRH3HRH2KDRALDH1A1
SCHEMBL1774550 0.83 HRH4 (1.00) HRH4HRH3HRH2KDR
SCHEMBL1776779 0.82 HRH4 (0.79) HRH4HRH3HRH2KDRCYP1A2
SCHEMBL1774487 0.80 HRH4 (0.72) HRH4HRH3HRH2KDRALDH1A1
SCHEMBL1774562 0.80 HRH4 (0.68) HRH4HRH3HRH2KDRALDH1A1
SCHEMBL1773934 0.80 HRH4 (0.68) HRH4HRH3HRH2KDR
SCHEMBL1775001 0.80 HRH4 (1.00) HRH4HRH3HRH2KDRCYP1A2
SCHEMBL1774691 0.77 HRH4 (0.67) HRH4HRH3HRH2KDR
SCHEMBL1775220 0.76 HRH4 (1.00) HRH4HRH3HRH2KDR
SCHEMBL1774962 0.75 HRH4 (0.67) HRH4HRH3HRH2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966162-A2 PYRIMIDINE DERIVATIVES Pfizer Limited (GB) 2008-09-10 EP disclosed
WO-2007072163-A2 PYRIMIDINE DERIVATIVES PFIZER LIMITED (GB) 2007-06-28 WO disclosed