SCHEMBL475258

SCHEMBL475258

CC(C)(C)OC(=O)N[C@H](C(=O)N1CCCC1C(=O)Nc1ccc(-c2[nH]c3ccc(NC(=O)[C@@H]4CCCN4C(=O)[C@H](NC(=O)OC(C)(C)C)c4ccccc4)cc3c2C(=O)O)cc1)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.62
CYP2C9 P11712 6/20 0.56
CYP2C19 P33261 6/20 0.56
CYP3A4 P08684 5/20 0.56
CYP2D6 P10635 2/20 0.56
CYP1A2 P05177 2/20 0.56
CMA1 P23946 7/20 0.42
NPC1 O15118 1/20 0.42
CTRC Q99895 4/20 0.42
JAK2 O60674 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 1/20 0.39
JAK3 P52333 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16291124 1.00 KCNH2 (0.62) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL20952254 1.00 KCNH2 (0.62) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL475256 1.00 KCNH2 (0.62) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL894917 0.94 KCNH2 (0.62) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL20952514 0.94 KCNH2 (0.62) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL24732245 0.94 KCNH2 (0.60) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL16290821 0.94 KCNH2 (0.62) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL10223689 0.93 KCNH2 (0.58) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL10222828 0.92 KCNH2 (0.58) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL16199243 0.92 KCNH2 (0.61) KCNH2CYP2C9CYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410844-A1 INHIBITORS OF HEPATITIS C VIRUS REPLICATION Merck Sharp & Dohme Corp. (US) 2012-02-01 EP claimed