SCHEMBL4752923

SCHEMBL4752923

CC(C)(C)OC(=O)N[C@H]1CCCC[C@@H]1n1cnc(C(=O)N2CCN(Cc3ccccc3)C[C@H]2Cc2ccccc2)c1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA4 P22748 2/20 0.40
CA9 Q16790 2/20 0.40
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ROCK1 Q13464 1/20 0.38
DPP4 P27487 2/20 0.35
DPP7 Q9UHL4 1/20 0.35
HDAC1 Q13547 1/20 0.35
CKS1B P61024 1/20 0.34
SKP1 P63208 1/20 0.34
SKP2 Q13309 1/20 0.34
AKT1 P31749 1/20 0.34
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
ACE P12821 1/20 0.34
NSD2 O96028 1/20 0.34
CCKAR P32238 1/20 0.34
CCKBR P32239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4752441 0.94 CA1 (0.36) CA1CA2CA4CA9KMT2A
SCHEMBL4752935 0.93 CA1 (0.43) CA1CA2CA4CA9ROCK1
SCHEMBL13705205 0.91 CA1 (0.41) CA1CA2CA4CA9L3MBTL1
SCHEMBL4752660 0.90 CA1 (0.40) CA1CA2CA4CA9ROCK1
SCHEMBL4293386 0.89 CA1 (0.45) CA1CA2CA4CA9ROCK1
SCHEMBL13705208 0.89 CA1 (0.41) CA1CA2CA4CA9L3MBTL1
SCHEMBL13705207 0.89 CA1 (0.39) CA1CA2CA4CA9L3MBTL1
SCHEMBL13705206 0.89 CA1 (0.39) CA1CA2CA4CA9KMT2A
SCHEMBL13705288 0.86 CA1 (0.38) CA1CA2CA4CA9ROCK1
SCHEMBL13705173 0.85 CA1 (0.36) CA1CA2CA4CA9L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed