SCHEMBL4754592

SCHEMBL4754592

Clc1nc(N2CCOCC2)c2cc(CN3CCC(N4CCOCC4)CC3)ccc2n1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.56
SMN1; SMN2 Q16637 1/20 0.47
PIK3CA P42336 12/20 0.46
MTOR P42345 12/20 0.46
PIK3CG P48736 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18032505 0.95 HRH3 (0.55) HRH3SMN1; SMN2PIK3CAMTORPIK3CG
SCHEMBL4752524 0.84 SMN1; SMN2 (0.52) HRH3SMN1; SMN2PIK3CAPIK3CG
SCHEMBL4789881 0.81 SMN1; SMN2 (0.43) HRH3SMN1; SMN2PIK3CAMTOR
SCHEMBL13982364 0.80 SMN1; SMN2 (0.48) HRH3SMN1; SMN2PIK3CAMTOR
SCHEMBL390035 0.78 PIK3CD (0.53) HRH3PIK3CAPIK3CG
SCHEMBL4754666 0.78 PIK3CA (0.65) PIK3CAMTORPIK3CG
SCHEMBL13982563 0.76 PIK3CA (0.52) PIK3CAMTORPIK3CG
SCHEMBL13982367 0.76 SMN1; SMN2 (0.42) SMN1; SMN2PIK3CAMTORPIK3CG
SCHEMBL3776763 0.74 SMN1; SMN2 (0.61) SMN1; SMN2PIK3CA
SCHEMBL996677 0.74 PIK3CD (0.56) HRH3PIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008152387-A1 QUINAZOLINE DERIVATIVES AS PI3 KINASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2008-12-18 WO disclosed