SCHEMBL4756397

SCHEMBL4756397

CC(c1ccccc1)N1CCN(c2c(Br)ncc3[nH]c(-c4ccc(CNC(=O)O)cc4)nc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 7/20 0.43
AURKA O14965 5/20 0.43
VSIR Q9H7M9 2/20 0.38
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
TRPC5 Q9UL62 1/20 0.37
KRAS P01116 1/20 0.36
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
ADORA2B P29275 1/20 0.36
PARP1 P09874 1/20 0.35
KDR P35968 1/20 0.34
AURKB Q96GD4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13985468 0.77 AURKA (0.41) DGAT1AURKAHDAC1TRPC5TNKS
SCHEMBL4789994 0.74 AURKA (0.43) AURKATRPC5TNKSTNKS2ADORA2B
SCHEMBL4789991 0.73 AURKA (0.47) AURKATRPC5ADORA2B
SCHEMBL209704 0.69 AURKA (0.53) AURKAHDAC4HDAC1PARP1
SCHEMBL208759 0.69 CHEK2 (0.40) DGAT1AURKAVSIRTNKSTNKS2
SCHEMBL208728 0.68 AURKA (0.47) AURKATRPC5TNKSTNKS2ADORA2B
SCHEMBL210610 0.68 MEN1 (0.43) DGAT1AURKATNKSTNKS2
SCHEMBL211374 0.67 AURKA (0.45) DGAT1AURKATRPC5KRASADORA2B
SCHEMBL4757469 0.67 AURKA (0.47) AURKAHDAC4HDAC1
SCHEMBL4790505 0.67 AURKA (0.54) AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed