SCHEMBL4758189

SCHEMBL4758189

C[C@@H](NC[C@H]1CN(CNc2ccc(C(=O)O)cc2Cl)C[C@@H]1c1ccccc1)c1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASR P41180 18/20 0.46
CYP2D6 P10635 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2B6 P20813 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4105924 0.85 CASR (0.46) CASRCYP2D6
SCHEMBL4105928 0.85 CASR (0.46) CASRCYP2D6
Hydrochloric Acid SCHEMBL4101551 0.82 CASR (0.53) CASRCYP2D6
Hydrochloric Acid SCHEMBL4101549 0.82 CASR (0.53) CASRCYP2D6
SCHEMBL1105843 0.82 CASR (0.45) CASRCYP2D6
SCHEMBL1105823 0.82 CASR (0.46) CASRCYP2D6
Hydrochloric Acid SCHEMBL4101450 0.82 CASR (0.55) CASRCYP2A6CYP2B6
Hydrochloric Acid SCHEMBL1096054 0.81 CASR (0.46) CASRCYP2D6
SCHEMBL4101477 0.79 CASR (0.53) CASRCYP2D6
SCHEMBL4105037 0.78 CASR (0.51) CASRCYP2D6CYP2A6CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1882684-A1 PYRROLIDINE DERIVATIVE OR SALT THEREOF Astellas Pharma Inc. (JP) 2008-01-30 EP disclosed