SCHEMBL4758320

SCHEMBL4758320

O/N=[C]/Cc1ccc(OCc2ccc(F)cc2F)nc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.40
AGXT P21549 2/20 0.40
MAOB P27338 1/20 0.40
ALKBH1 Q13686 1/20 0.37
CCR5 P51681 1/20 0.37
GSK3B P49841 2/20 0.37
BACE1 P56817 2/20 0.37
PPARA Q07869 1/20 0.36
MAPK14 Q16539 9/20 0.35
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
PTGER1 P34995 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758323 1.00 IDO1 (0.40) IDO1AGXTMAOBALKBH1CCR5
SCHEMBL510480 0.81 IDO1 (0.38) IDO1AGXTMAOBALKBH1CCR5
SCHEMBL510479 0.81 IDO1 (0.38) IDO1AGXTMAOBALKBH1CCR5
SCHEMBL4757964 0.75 EGLN1 (0.42) MAOB
SCHEMBL4757966 0.75 EGLN1 (0.42) MAOB
SCHEMBL2942352 0.69 NPC1 (0.38) AGXTMAOB
SCHEMBL2942355 0.69 NPC1 (0.38) AGXTMAOB
SCHEMBL29975341 0.68 GRM5 (0.53) IDO1AGXTMAOBMAPK14
SCHEMBL28678965 0.67 MIF (0.42) IDO1AGXT
SCHEMBL1711843 0.66 IDO1 (0.47) IDO1AGXTMAOBALKBH1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1944303-B1 PYRIDINE DERIVATIVE SUBSTITUTED BY HETEROCYCLE AND FUNGICIDE CONTAINING THE SAME EISAI R&D MAN CO LTD (JP) 2013-08-21 EP disclosed
EP-1944303-A1 PYRIDINE DERIVATIVE SUBSTITUTED BY HETEROCYCLE AND FUNGICIDE CONTAINING THE SAME Eisai R&D Management Co., Ltd. (JP) 2008-07-16 EP disclosed