SCHEMBL4758624

SCHEMBL4758624

CN1CCN(c2ccc(N/C=C3/C(=O)Nc4cc(C(=O)c5cccc(NC(=O)Nc6ccc(Cl)cc6)c5)ccc43)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 3/20 0.54
FLT3 P36888 5/20 0.46
KDR P35968 3/20 0.46
FLT4 P35916 2/20 0.46
KIT P10721 1/20 0.46
NTRK1 P04629 3/20 0.45
NTRK3 Q16288 1/20 0.45
CNR1 P21554 3/20 0.44
AURKB Q96GD4 1/20 0.44
NTRK2 Q16620 3/20 0.43
F10 P00742 2/20 0.42
AURKA O14965 1/20 0.42
CNR2 P34972 1/20 0.42
TNKS O95271 1/20 0.41
PARP1 P09874 1/20 0.41
PARP14 Q460N5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703897 1.00 CSF1R (0.54) CSF1RFLT3KDRFLT4KIT
SCHEMBL4758071 0.95 CSF1R (0.52) CSF1RFLT3KDRFLT4KIT
SCHEMBL4706778 0.95 CSF1R (0.52) CSF1RFLT3KDRFLT4KIT
SCHEMBL4759327 0.94 CSF1R (0.56) CSF1RFLT3KDRFLT4KIT
SCHEMBL4703036 0.94 CSF1R (0.56) CSF1RFLT3KDRFLT4KIT
SCHEMBL4757095 0.94 NTRK1 (0.50) CSF1RFLT3NTRK1NTRK3AURKB
SCHEMBL4757094 0.94 NTRK1 (0.50) CSF1RFLT3NTRK1NTRK3AURKB
SCHEMBL4755255 0.93 CSF1R (0.54) CSF1RFLT3KDRFLT4KIT
SCHEMBL4755254 0.93 CSF1R (0.54) CSF1RFLT3KDRFLT4KIT
SCHEMBL4757149 0.92 CSF1R (0.53) CSF1RFLT3KDRFLT4KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902025-A1 KINASE INHIBITORS Allergan, Inc. (US) 2008-03-26 EP claimed
US-20070032478-A1 Kinase Inhibitors ALLERGAN, INC. 2007-02-08 US claimed
WO-2007008895-A1 KINASE INHIBITORS ALLERGAN, INC. (US) 2007-01-18 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070032478-A1 Kinase Inhibitors ABL1, LCK, ERBB2 CSF1R 877/4885FLT3 87/4885KDR 226/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.