SCHEMBL4760934

SCHEMBL4760934

CCC(=O)NCCn1cc(C(=O)N2CCN(c3ccccc3F)CC2)c2ccc(Cl)cc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
PPARG P37231 1/20 0.50
NCOA2 Q15596 1/20 0.50
NCOA1 Q15788 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
PIK3CD O00329 1/20 0.46
PIK3R1 P27986 1/20 0.46
PIK3CA P42336 1/20 0.46
PIK3CG P48736 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
TSHR P16473 1/20 0.46
TP53 P04637 2/20 0.46
AVPR1A P37288 3/20 0.45
CNR1 P21554 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL613390 0.91 SMN1; SMN2 (0.47) USP2CYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL615559 0.88 SMN1; SMN2 (0.45) USP2CYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL613549 0.88 TP53 (0.47) USP2PIK3CDPIK3R1PIK3CAPIK3CG
SCHEMBL615054 0.86 AVPR1A (0.51) USP2CYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL615567 0.86 SMN1; SMN2 (0.53) USP2CYP1A2CYP2C19NPSR1PIK3CD
SCHEMBL613033 0.85 AVPR1A (0.51) USP2CYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL615036 0.85 TP53 (0.45) USP2PIK3CDPIK3R1PIK3CAPIK3CG
SCHEMBL613100 0.84 AVPR1A (0.63) USP2CYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL614430 0.84 AVPR1A (0.60) USP2NPSR1PIK3CDPIK3R1PIK3CA
SCHEMBL613537 0.84 SMN1; SMN2 (0.49) USP2NPSR1PIK3CDPIK3R1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917255-A2 INDOL-3-YL-CARBONYL-PIPERIDIN AND PIPERAZIN DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-05-07 EP disclosed
WO-2007014851-A2 INDOL-3-YL-CARBONYL-PIPERIDIN AND PIPERAZIN DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-02-08 WO disclosed