SCHEMBL4761565

SCHEMBL4761565

Nc1ccc(-c2ccccc2)cc1NC(=O)c1cc2ccc(C3(C4CCC5(CCCN5)CC4)CCC4(CCCN4)CC3)cc2s1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 16/20 0.53
HDAC3 O15379 12/20 0.53
KCNH2 Q12809 6/20 0.53
HDAC2 Q92769 7/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4760696 0.76 HDAC1 (0.70) HDAC1HDAC3KCNH2HDAC2
SCHEMBL4721527 0.73 HDAC1 (0.54) HDAC1HDAC3KCNH2HDAC2
SCHEMBL5330808 0.72 HDAC1 (0.68) HDAC1HDAC3KCNH2HDAC2
SCHEMBL1641006 0.69 HDAC2 (0.61) HDAC1HDAC3KCNH2HDAC2
SCHEMBL1640200 0.69 HDAC1 (1.00) HDAC1HDAC3KCNH2HDAC2
SCHEMBL1640304 0.69 HDAC1 (0.80) HDAC1HDAC3KCNH2HDAC2
SCHEMBL12727254 0.67 HDAC1 (0.65) HDAC1HDAC3KCNH2HDAC2
SCHEMBL1639796 0.67 HDAC1 (1.00) HDAC1HDAC3KCNH2HDAC2
SCHEMBL4580299 0.67 HDAC2 (0.56) HDAC1HDAC3HDAC2
SCHEMBL1640675 0.66 KCNH2 (0.74) HDAC1HDAC3KCNH2HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954698-A1 SPIROCYCLIC COMPOUNDS AS HDAC INHIBITORS Merck & Co., Inc. (US) 2008-08-13 EP claimed
WO-2007061880-A1 SPIROCYCLIC COMPOUNDS AS HDAC INHIBITORS MERCK & CO., INC. (US) 2007-05-31 WO claimed