SCHEMBL4762779

SCHEMBL4762779

CC(C)(C)C(F)(F)c1cccc(Oc2ccc(Nc3ncnc4ccn(CCN)c34)cc2Cl)c1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.72
ERBB2 P04626 20/20 0.72
ERBB3 P21860 16/20 0.72
ERBB4 Q15303 16/20 0.72
BMPR1B O00238 1/20 0.67
EPHB6 O15197 1/20 0.67
LCK P06239 1/20 0.67
LYN P07948 1/20 0.67
MET P08581 1/20 0.67
CSK P41240 1/20 0.67
MAP2K1 Q02750 1/20 0.67
MAP2K5 Q13163 1/20 0.67
AURKB Q96GD4 1/20 0.67
NLK Q9UBE8 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3510098 0.99 EGFR (0.71) EGFRERBB2ERBB3ERBB4BMPR1B
SCHEMBL3506027 0.92 EGFR (0.85) EGFRERBB2ERBB3ERBB4BMPR1B
SCHEMBL3127092 0.92 EGFR (0.85) EGFRERBB2ERBB3ERBB4BMPR1B
Hydrochloric Acid SCHEMBL2748120 0.91 EGFR (0.83) EGFRERBB2ERBB3ERBB4BMPR1B
SCHEMBL3506249 0.89 EGFR (0.86) EGFRERBB2ERBB3ERBB4BMPR1B
SCHEMBL3505151 0.87 EGFR (0.88) EGFRERBB2ERBB3ERBB4BMPR1B
SCHEMBL5141834 0.87 EGFR (0.85) EGFRERBB2ERBB3ERBB4BMPR1B
Hydrochloric Acid SCHEMBL2747039 0.86 EGFR (0.83) EGFRERBB2ERBB3ERBB4BMPR1B
SCHEMBL13226160 0.86 EGFR (0.90) EGFRERBB2ERBB3ERBB4BMPR1B
SCHEMBL3505490 0.86 EGFR (0.69) EGFRERBB2ERBB3ERBB4BMPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957495-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-08-20 EP disclosed
WO-2007064045-A1 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-06-07 WO disclosed