SCHEMBL4763459

SCHEMBL4763459

O=C(O)NCCn1ccc2ncnc(Nc3ccc4c(ccn4Cc4ccccn4)c3)c21

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 14/20 0.56
EGFR P00533 13/20 0.56
ERBB4 Q15303 4/20 0.56
ERBB3 P21860 1/20 0.42
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3505760 0.88 ERBB2 (0.55) ERBB2EGFRERBB4ERBB3
SCHEMBL4761967 0.87 ERBB2 (0.56) ERBB2EGFRERBB4KCNH2
Hydrochloric Acid SCHEMBL3507866 0.86 EGFR (0.53) ERBB2EGFRERBB4ERBB3KCNH2
SCHEMBL3507874 0.85 ERBB2 (0.53) ERBB2EGFRERBB4ERBB3KCNH2
SCHEMBL27751027 0.85 ERBB2 (0.55) ERBB2EGFRERBB4KCNH2
SCHEMBL2749154 0.81 ERBB2 (0.58) ERBB2EGFRERBB4ERBB3KCNH2
SCHEMBL14494991 0.77 EGFR (0.47) ERBB2EGFRERBB4ERBB3
SCHEMBL4194347 0.77 ERBB2 (0.56) ERBB2EGFRERBB4KCNH2
SCHEMBL3618270 0.75 ERBB2 (0.56) ERBB2EGFRERBB4KCNH2
SCHEMBL4197751 0.75 ERBB2 (0.69) ERBB2EGFRERBB4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957495-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-08-20 EP disclosed
WO-2007064045-A1 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-06-07 WO disclosed