SCHEMBL4765978

SCHEMBL4765978

N=C(N)NCCCCNc1cc(-c2cccnc2)nc(-c2ccccn2)n1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.44
HDAC6 Q9UBN7 11/20 0.44
CYP2A6 P11509 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
ROS1 P08922 3/20 0.43
SLC2A1 P11166 1/20 0.42
ABL1 P00519 1/20 0.42
BCR P11274 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771962 0.83 HDAC1 (0.44) HDAC1HDAC6CYP2A6CYP3A4CYP2C9
SCHEMBL4771979 0.83 HDAC1 (0.44) HDAC1HDAC6CYP2A6CYP3A4CYP2C9
SCHEMBL2238098 0.79 PTGDR (0.53) CYP2A6CYP3A4CYP2C9SLC2A1
SCHEMBL2240945 0.79 GBA1 (0.54) CYP2A6CYP3A4CYP2C9SLC2A1
SCHEMBL2237295 0.78 CYP2A6 (0.45) HDAC1CYP2A6CYP3A4CYP2C9SLC2A1
SCHEMBL2242475 0.78 PTGDR (0.54) CYP2A6CYP3A4CYP2C9SLC2A1
SCHEMBL3630638 0.77 SMN1; SMN2 (0.55) ABL1BCR
SCHEMBL2237320 0.77 HIF1A (0.47) HDAC1CYP2A6CYP3A4CYP2C9SLC2A1
SCHEMBL4777383 0.77 METAP1 (0.47) HDAC1HDAC6CYP3A4CYP2C9ROS1
SCHEMBL4769037 0.77 GSK3A (0.43) HDAC1HDAC6CYP2A6CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed