SCHEMBL4766752

SCHEMBL4766752

CC(C)c1cc(C(=O)N2CCN(CC=O)CC2)c(O)cc1O

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 19/20 0.62
HSP90AB1 P08238 6/20 0.62
HSP90B1 P14625 4/20 0.53
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL487620 0.81 HSP90AA1 (0.72) HSP90AA1HSP90AB1HSP90B1
SCHEMBL487588 0.81 HSP90AA1 (0.72) HSP90AA1HSP90AB1HSP90B1
SCHEMBL487987 0.80 HSP90AA1 (0.60) HSP90AA1HSP90AB1HSP90B1
SCHEMBL2948707 0.80 HSP90AA1 (0.60) HSP90AA1HSP90AB1HSP90B1HDAC8
SCHEMBL487667 0.77 HSP90AA1 (1.00) HSP90AA1HSP90AB1HSP90B1
SCHEMBL10256000 0.76 HSP90AA1 (0.61) HSP90AA1HSP90AB1HSP90B1HDAC8
SCHEMBL15000795 0.76 HSP90AA1 (0.68) HSP90AA1HSP90AB1HSP90B1
SCHEMBL10256275 0.76 HSP90AA1 (0.68) HSP90AA1HSP90AB1HSP90B1
SCHEMBL488032 0.75 HSP90AA1 (0.64) HSP90AA1HSP90AB1HSP90B1HDAC8
SCHEMBL2948708 0.75 HSP90AA1 (0.60) HSP90AA1HSP90AB1HSP90B1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1883402-A2 HYDROXYBENZAMIDE DERIVATIVES AND THEIR USE AS INHIBITORS OF HSP90 Astex Therapeutics Limited (GB) 2008-02-06 EP disclosed
WO-2006109075-A2 HYDROXYBENZAMIDE DERIVATIVES AND THEIR USE AS INHIBITORS OF HSP90 ASTEX THERAPEUTICS LIMITED (GB) 2006-10-19 WO disclosed