SCHEMBL4767463

SCHEMBL4767463

O=c1c([N+](=O)[O-])c(/C=C/c2cnn(-c3ccccc3)c2)n(C2CCC2)c(=O)n1C1CCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MTOR P42345 2/20 0.36
ACKR3 P25106 1/20 0.36
RPTOR Q8N122 1/20 0.35
MLST8 Q9BVC4 1/20 0.35
HSP90AA1 P07900 1/20 0.35
GRM1 Q13255 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
MITF O75030 1/20 0.34
ALDH1A1 P00352 6/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
NPSR1 Q6W5P4 3/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4767470 1.00 NPC1 (0.41) NPC1RAB9ASMN1; SMN2MTORACKR3
SCHEMBL4792631 0.87 NPC1 (0.35) NPC1RAB9ASMN1; SMN2MTORACKR3
SCHEMBL4792628 0.87 NPC1 (0.35) NPC1RAB9ASMN1; SMN2MTORACKR3
SCHEMBL4792629 0.87 SMN1; SMN2 (0.35) NPC1RAB9ASMN1; SMN2MTORACKR3
SCHEMBL4769797 0.86 PDE4A (0.37) NPC1RAB9ASMN1; SMN2MTORACKR3
SCHEMBL4769812 0.86 PDE4A (0.37) NPC1RAB9ASMN1; SMN2MTORACKR3
SCHEMBL4858967 0.80 HSP90AA1 (0.44) MTORHSP90AA1GRM1ALDH1A1MEN1
SCHEMBL4769541 0.79 MAPT (0.37) HDAC2MITFALDH1A1MAPTPKM
SCHEMBL4769532 0.79 MAPT (0.37) HDAC2MITFALDH1A1MAPTPKM
SCHEMBL4762674 0.78 ADORA2A (0.36) ALDH1A1KDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed