SCHEMBL4769964

SCHEMBL4769964

CNCC(C)c1ccc(-n2cc3cccc(C(N)=O)c3n2)cc1

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.74
PARP2 Q9UGN5 11/20 0.74
PARP3 Q9Y6F1 11/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21122508 0.88 PARP1 (0.72) PARP1PARP2PARP3
SCHEMBL20757943 0.86 PARP1 (0.69) PARP1PARP2PARP3
SCHEMBL2263902 0.85 PARP1 (1.00) PARP1PARP2PARP3
SCHEMBL21122507 0.85 PARP1 (0.78) PARP1PARP2PARP3
Hydrochloric Acid SCHEMBL2264068 0.84 PARP1 (0.98) PARP1PARP2PARP3
Hydrochloric Acid SCHEMBL2267815 0.84 PARP1 (0.98) PARP1PARP2PARP3
Hydrochloric Acid SCHEMBL2264646 0.84 PARP1 (0.98) PARP1PARP2PARP3
SCHEMBL2265179 0.82 PARP1 (1.00) PARP1PARP2PARP3
Hydrochloric Acid SCHEMBL2267601 0.81 PARP1 (0.98) PARP1PARP2PARP3
SCHEMBL4769970 0.80 PARP1 (0.72) PARP1PARP2PARP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007733-A1 AMIDE SUBSTITUTED INDAZOLE AND BENZOTRIAZOLE DERIVATIVES AS POLY(ADP-RIBOSE)POLYMERASE (PARP) INHIBITORS Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2008-12-31 EP disclosed
WO-2007113596-A1 AMIDE SUBSTITUTED INDAZOLE AND BENZOTRIAZOLE DERIVATIVES AS POLY(ADP-RIBOSE)POLYMERASE (PARP) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-10-11 WO disclosed