SCHEMBL4771978

SCHEMBL4771978

NS(=O)(=O)c1ccc(CCNc2cc(-c3cccnc3)nc(-c3ccccn3)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 3/20 0.51
FYN P06241 1/20 0.51
TDP1 Q9NUW8 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
RXFP1 Q9HBX9 2/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
CA2 P00918 4/20 0.46
CA9 Q16790 4/20 0.46
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA14 Q9ULX7 1/20 0.46
KCNH2 Q12809 1/20 0.46
MRGPRX1 Q96LB2 1/20 0.45
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
PIM1 P11309 1/20 0.43
PTGS2 P35354 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768768 0.90 PTGDR (0.53) PTGDRALDH1A1CYP3A4CYP2C9PTGS2
SCHEMBL2242475 0.86 PTGDR (0.54) PTGDRTDP1KMT2AKDM4EALDH1A1
SCHEMBL2238098 0.86 PTGDR (0.53) PTGDRTDP1KMT2AKDM4EALDH1A1
SCHEMBL2237693 0.83 PTGDR (0.73) PTGDRKMT2A
SCHEMBL2240945 0.81 GBA1 (0.54) PTGDRALDH1A1CYP3A4CYP2C9MAPT
SCHEMBL2239971 0.81 SMN1; SMN2 (0.53) PTGDRMEN1KMT2AKDM4EALDH1A1
SCHEMBL2237295 0.80 CYP2A6 (0.45) PTGDRKDM4EALDH1A1KCNH2CYP3A4
SCHEMBL2237320 0.80 HIF1A (0.47) PTGDRKDM4EALDH1A1KCNH2CYP3A4
SCHEMBL2238820 0.80 PTGDR (0.48) PTGDRKDM4EALDH1A1KCNH2CYP3A4
SCHEMBL2241291 0.80 KMT2A (0.46) PTGDRTDP1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed