SCHEMBL4772610

SCHEMBL4772610

CCCCn1c(-c2ccccc2)nc(-c2ccccc2)c1CN(Cc1cc(F)ccc1F)Cc1ccccc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 1/20 0.41
BCHE P06276 7/20 0.39
ACHE P22303 6/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
TACR1 P25103 1/20 0.38
CASR P41180 1/20 0.38
TSHR P16473 2/20 0.37
MAOB P27338 3/20 0.37
CHRNE Q04844 1/20 0.37
TP53 P04637 2/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PKM P14618 1/20 0.36
MAPT P10636 1/20 0.36
GNRHR P30968 1/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135688 0.90 C5AR1 (0.45) C5AR1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL4769336 0.90 C5AR1 (0.43) C5AR1BCHEALDH1A1KDM4ELMNA
SCHEMBL5134844 0.89 C5AR1 (0.44) C5AR1ALDH1A1KDM4ETSHRGNRHR
SCHEMBL5074353 0.89 C5AR1 (0.44) C5AR1BCHEACHEALDH1A1KDM4E
SCHEMBL5135193 0.88 BCHE (0.43) C5AR1BCHEACHETACR1CASR
SCHEMBL5069962 0.88 BCHE (0.45) C5AR1BCHEACHETACR1CASR
SCHEMBL5137131 0.86 C5AR1 (0.41) C5AR1ALDH1A1KDM4ETSHRTP53
SCHEMBL5134673 0.85 C5AR1 (0.43) C5AR1BCHEACHEALDH1A1KDM4E
SCHEMBL5135095 0.85 BCHE (0.47) C5AR1BCHEACHEMAOBTP53
SCHEMBL5137586 0.85 C5AR1 (0.40) C5AR1ALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322309-B1 HIGH AFFINITY SMALL MOLECULE C5A RECEPTOR MODULATORS NEUROGEN CORP (US) 2008-08-13 EP claimed