SCHEMBL4773440

SCHEMBL4773440

Nc1cc(-c2cccnc2)nc(-c2ccccn2)n1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.63
NPC1 O15118 1/20 0.56
TP53 P04637 1/20 0.56
PKM P14618 1/20 0.56
TSHR P16473 1/20 0.56
RAB9A P51151 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
CYP19A1 P11511 2/20 0.51
KDM4E B2RXH2 3/20 0.50
ADORA2A P29274 1/20 0.50
ADORA1 P30542 1/20 0.50
ALOX15 P16050 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
F2 P00734 1/20 0.49
F12 P00748 1/20 0.49
HSP90AA1 P07900 1/20 0.49
HSP90AB1 P08238 1/20 0.49
PTK2 Q05397 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
GRM5 P41594 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7264634 0.86 ADORA2A (0.68) NPC1TP53PKMTSHRRAB9A
SCHEMBL4768766 0.85 CYP2A6 (0.46) CYP2A6NPC1TP53PKMTSHR
SCHEMBL24589930 0.85 CYP2A6 (0.67) CYP2A6NPC1TP53PKMTSHR
SCHEMBL13912521 0.84 ADORA2A (0.71) CYP2A6NPC1TP53TSHRRAB9A
SCHEMBL19830922 0.84 ADORA2A (0.59) CYP2A6TP53TSHRSMN1; SMN2CYP19A1
SCHEMBL2239691 0.82 CYP2A6 (0.63) CYP2A6NPC1TP53PKMTSHR
SCHEMBL19047219 0.82 CYP2A6 (0.63) CYP2A6NPC1TP53PKMTSHR
SCHEMBL4773465 0.82 CYP2A6 (0.63) CYP2A6NPC1TP53PKMTSHR
SCHEMBL19054158 0.81 ADORA2A (0.71) CYP2A6NPC1TP53TSHRRAB9A
SCHEMBL16606290 0.81 CYP2A6 (0.70) CYP2A6NPC1TP53PKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed