SCHEMBL4773661

SCHEMBL4773661

CC(C)COC(=O)N1C(C(=O)N[C@@H](CC(C)C)C(=O)NCCCCNS(=O)(=O)c2ccc(F)cc2Cl)CC2CCCCC21

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 2/20 0.43
F2 P00734 3/20 0.40
PRSS1 P07477 3/20 0.38
PRSS2 P07478 3/20 0.38
PRSS3 P35030 3/20 0.38
BMP1 P13497 1/20 0.37
NMUR2 Q9GZQ4 1/20 0.37
NMUR1 Q9HB89 1/20 0.37
ELANE P08246 2/20 0.35
CCR1 P32246 1/20 0.35
ADAM17 P78536 1/20 0.35
CTSL P07711 3/20 0.35
TRPV4 Q9HBA0 1/20 0.35
CTSB P07858 2/20 0.34
CTSS P25774 2/20 0.34
CTSK P43235 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4140140 0.92 CAPN1 (0.43) CAPN1F2PRSS1PRSS2PRSS3
SCHEMBL4136304 0.82 CAPN1 (0.53) CAPN1BMP1CCR1ADAM17CTSL
SCHEMBL5434636 0.80 CAPN1 (0.51) CAPN1BMP1CCR1ADAM17CTSL
SCHEMBL4777748 0.80 CAPN1 (0.40) CAPN1BMP1CCR1ADAM17CTSL
SCHEMBL4139968 0.79 CAPN1 (0.44) CAPN1BMP1CCR1ADAM17CTSL
SCHEMBL4140823 0.79 CAPN1 (0.46) CAPN1BMP1CCR1ADAM17CTSL
SCHEMBL4141710 0.78 CAPN1 (0.49) CAPN1BMP1CCR1ADAM17CTSL
SCHEMBL4141985 0.78 CAPN1 (0.46) CAPN1BMP1CCR1ADAM17CTSL
SCHEMBL4142973 0.78 CAPN1 (0.48) CAPN1BMP1CCR1ADAM17CTSL
SCHEMBL4130820 0.77 CAPN1 (0.47) CAPN1BMP1CCR1ADAM17CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940785-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SmithKline Beecham Corporation (US) 2008-07-09 EP claimed
WO-2007030761-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO claimed