SCHEMBL4773985

SCHEMBL4773985

Brc1cc2c(c(-c3ccc4ncnc(NC5CCCCC5)c4c3)c1)OCC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD38 P28907 4/20 0.51
CYP1A2 P05177 9/20 0.48
CYP3A4 P08684 8/20 0.48
CYP2D6 P10635 7/20 0.48
CYP2C19 P33261 7/20 0.48
CLK4 Q9HAZ1 7/20 0.48
USP2 O75604 6/20 0.48
LMNA P02545 6/20 0.48
TSHR P16473 4/20 0.48
MAP4K4 O95819 1/20 0.48
HSD17B10 Q99714 4/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPK1 P28482 2/20 0.47
ALDH1A1 P00352 1/20 0.47
ALOX15 P16050 1/20 0.47
IRAK4 Q9NWZ3 4/20 0.47
DYRK1A Q13627 1/20 0.46
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359186 0.85 PDE5A (0.35) CD38CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4353426 0.77 HTT (0.43) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL4357479 0.76 IRAK4 (0.75) CD38CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4353446 0.75 IRAK4 (0.77) CD38CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4358072 0.71 CD38 (0.64) CD38CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4351313 0.71 MAP4K4 (0.74) CD38CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4355129 0.71 DYRK1A (0.33) CYP1A2DYRK1A
SCHEMBL21318842 0.70 IRAK4 (0.73) CD38CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL17665803 0.70 CD38 (0.63) CD38CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4355227 0.70 CYP1A2 (0.67) CD38CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009078-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed